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EAAT2 activator 1
CAS No. 892415-28-0
EAAT2 activator 1( F2005-0304 | 3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine )
Catalog No. M28620 CAS No. 892415-28-0
F2005-0304 is a thiopyridazine derivative that has been found to increase EAAT2 protein levels in astrocytes.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 31 | Get Quote |
|
| 5MG | 50 | Get Quote |
|
| 10MG | 87 | Get Quote |
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| 25MG | 178 | Get Quote |
|
| 50MG | 330 | Get Quote |
|
| 100MG | 491 | Get Quote |
|
| 500MG | 1071 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameEAAT2 activator 1
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NoteResearch use only, not for human use.
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Brief DescriptionF2005-0304 is a thiopyridazine derivative that has been found to increase EAAT2 protein levels in astrocytes.
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DescriptionF2005-0304 is a thiopyridazine derivative that has been found to increase EAAT2 protein levels in astrocytes.
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In Vitro——
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In Vivo——
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SynonymsF2005-0304 | 3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine
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PathwayOthers
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TargetOther Targets
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RecptorBD1-BRD4|BRD4-BD2
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Research Area——
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Indication——
Chemical Information
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CAS Number892415-28-0
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Formula Weight331.8
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Molecular FormulaC16H11ClFN3S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 25 mg/mL (75.35 mM)
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SMILESFc1cccc(Cl)c1CSc(cc1)nnc1-c1ncccc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Kharenko OA, et al. Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain (BET) Inhibitors Targeting a Methionine. J Med Chem. 2018 Sep 27;61(18):8202-8211.
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